NIGERIAN JOURNAL OF SCIENCE AND ENVIRONMENT
Journal of the Faculties of Science and Agriculture, Delta State University, Abraka, Nigeria

ISSN: 1119-9008
DOI: 10.5987/UJ-NJSE
Email: njse@universityjournals.org


EFFECT OF METHANOL EXTRACT OF NEWBOULDIA LAEVIS STEM BARK ON THE UTERUS OF NON-PREGNANT RATS

DOI: 10.5987/UJ-NJSE.16.016.2   |   Article Number: 8559E616   |   Vol.12 (2) - September 2013

Authors:  Ayinde B.A and Owolabi O.J

Keywords: Oxytocin, Uterus, Herbal medicine, Tocolytic, Antagonism

The plant Newbouldia laevis NEEM (P. Beauv), Bignoniaceae family is locally used in Nigeria for

contracting the uterus to facilitate delivery. The stem bark was extracted using methanol via maceration

and its effect on the uterus investigated. The effects of both the crude extract (0.8mg/ml)

and the aqueous fraction on the uterus were examined against oxytocin (0.04-1.6x10-2) and acetylcholine

(0.04-16 mg/ml) induced contractions. A significant reduction was noted in the force of

contraction in the presence of the extract such that 0.51+ 0.12g produced by 0.04x10-2 oxytocin

was significantly (p<0.0001) reduced to 0.059+0.013g in the presence of the extract. The aqueous

fraction was observed to produce similar effects though not as significant as the crude extract. The

aqueous fraction of the extract remarkably inhibited (p<0.05) acetylcholine induced contractions at

all concentrations tested. The effect of both the crude extract and its aqueous fraction were comparable

with those of salbutamol and atropine on oxytocin and acetylcholine induced contractions

respectively. The phytochemical screening revealed the presence of alkaloids, saponins, tannins

and flavonoids. In conclusion as opposed to the oxytocic effect claimed in ethno medicine, a tocolytic

effect was observed. This effect may be mediated either via blockade of oxytocic receptors or

muscarinic receptor blockade. Saponins and tannins may also contribute to its relaxant effect on a

non-pregnant uterus.

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